William N. Setzer

Pharmaceuticals from Zimbabwean Traditional Herbal Medicine

The long term objectives of this project is discovery of new anti-infective and antitumor agents using traditional Zimbabwean ethnopharmacology as a guide. This project will involve collection of plant materials which already have a history of applications in the traditional medicine of the Ndebele people from Matabeleland, Zimbabwe. We will concentrate on plants which show promise for anti-infective activity (i.e., those used traditionally for treatment of wounds, skin diseases, venereal disease, infections, etc.), but which have not been examined phytochemically. Plant materials will be extracted and the crude extracts screened for biological activity (antimicrobial and cytotoxic). Extracts which show promising bioactivity will be subjected to activity-directed chromatographic separation in order to isolate and purify the active components. The active materials will be identified using spectroscopic and crystallographic techniques. This research provides an excellent opportunity to identify novel phytochemical agents which could serve to combat emerging infectious diseases, opportunistic or drug resistant microorganisms and tumors.

An especially attractive feature of this project is the interdisciplinary and interinstitutional character of the research. The proposed research involves an unprecidented collaboration between investigators from all three institutions of higher education in Huntsville, Alabama: the historically black/Seventh Day Adventist Oakwood College, historically black Alabama A & M University, and the University of Alabama in Huntsville. The collaboration provides opportunities for interaction between faculty members and student researchers, and allows greater access to different facilities from the three participating campuses. In addition, the collaboration with the University of Zimbabwe brings unique access to the phytochemical and ethnobotanical riches of Matabeleland, Zimbabwe. This research project provides excellent hands-on experiences for undergraduate students from three different institutions which already have a tradition in quality undergraduate scientific education.